GPCR screening

GPCR Screening & Profiling Assays

SB offers a broad selection of radioligand binding & cell based GPCR assays with fast turnaround times to enhance your discovery research. From high throughput screening to routine hit-to-lead optimization and selectivity profiling, SB's flexible services can be adapted to meet the most demading timelines.

GPCR targets

Target Radioligand Binding Cell-Based
5HTR1A Green Dot Green Dot
5HTR1B   Green Dot
5HTR2A Green Dot Green Dot
5HTR2B   Green Dot
5HTR2C Green Dot  
5HTR6 Green Dot  
5HTR7 Green Dot  
AdoR A1 Green Dot Green Dot
AdoR A2a Green Dot Green Dot
AdoR A2b Green Dot Green Dot
AdoR A3   Green Dot
ADRA1A Green Dot Green Dot
ADRA1B Green Dot  
ADRA2A Green Dot Green Dot
ADRA2C Green Dot  
ADRB1   Green Dot
ADRB2   Green Dot
BDKRB2   Green Dot
CHRM1 Green Dot Green Dot
CHRM2 Green Dot Green Dot
CHRM3 Green Dot Green Dot
CHRM4 Green Dot Green Dot
CHRM5 Green Dot Green Dot
CNR1 Green Dot Green Dot
CNR2 Green Dot Green Dot
CCKAR   Green Dot
DRD1 Green Dot Green Dot
DRD2 Green Dot Green Dot
DRD3 Green Dot  
DRD4 Green Dot  
EDNRA   Green Dot
F2RL1   Green Dot
F2RL3   Green Dot
HRH1   Green Dot
HRH2   Green Dot
OPRD1   Green Dot
OPRK1   Green Dot
OPRM1   Green Dot
P2RY2   Green Dot
SMO Green Dot  
VPR1A   Green Dot

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